GABA transporter

GABA transporters (gamma-aminobutyric acid transporters) are a family of neurotransmitter / sodium symporters, belonging to the solute carrier 6 (SLC6) family.[1][2] They are found in various regions of the brain in different cell types, such as neurons and astrocytes.

These transporters are primarily responsible for the regulation of extracellular GABA concentration during basal and synaptic activity. They are responsible for creating a GABA gradient which is determined by the membrane potential, and the concentration of Na+ and Cl. They are also present on the plasma membrane of neurons and glia which help define their function of regulation of GABA concentration as they act as the receptors that facilitate recycling of GABA in the extracellular space.[1] GABA transporters are a common target for anticonvulsant drugs against seizure disorders such as epilepsy.[3]

  1. ^ a b Scimemi, A (2014-06-17). "Structure, function, and plasticity of GABA transporters". Frontiers in Cellular Neuroscience. 8: 161. doi:10.3389/fncel.2014.00161. PMC 4060055. PMID 24987330.
  2. ^ Bernstein EM, Quick MW (January 1999). "Regulation of gamma-aminobutyric acid (GABA) transporters by extracellular GABA". The Journal of Biological Chemistry. 274 (2): 889–95. doi:10.1074/jbc.274.2.889. PMID 9873028.
  3. ^ Richerson GB, Wu Y (2004). "Role of the GABA Transporter in Epilepsy". Recent Advances in Epilepsy Research. Advances in Experimental Medicine and Biology. Vol. 548. Springer US. pp. 76–91. doi:10.1007/978-1-4757-6376-8_6. ISBN 9781441934185. PMID 15250587.