Ryanodine-Inositol 1,4,5-triphosphate receptor calcium channels

Ryanodine receptor 2
Identifiers
SymbolRYR2
PfamPF02026
InterProIPR003032
SMARTSM00054
PROSITEPS50188
TCDB1.A.3
OPM superfamily8
OPM protein6dr2
Available protein structures:
Pfam  structures / ECOD  
PDBRCSB PDB; PDBe; PDBj
PDBsumstructure summary
PDB4JKQ

The ryanodine-inositol 1,4,5-triphosphate receptor Ca2+ channel (RIR-CaC) family includes Ryanodine receptors and Inositol trisphosphate receptors. Members of this family are large proteins, some exceeding 5000 amino acyl residues in length. This family belongs to the Voltage-gated ion channel (VIC) superfamily. Ry receptors occur primarily in muscle cell sarcoplasmic reticular (SR) membranes, and IP3 receptors occur primarily in brain cell endoplasmic reticular (ER) membranes where they effect release of Ca2+ into the cytoplasm upon activation (opening) of the channel. They are redox sensors, possibly providing a partial explanation for how they control cytoplasmic Ca2+. Ry receptors have been identified in heart mitochondria where they provide the main pathway for Ca2+ entry.[1] Sun et al. (2011) have demonstrated oxygen-coupled redox regulation of the skeletal muscle ryanodine receptor-Ca2+ release channel (RyR1;TC# 1.A.3.1.2) by NADPH oxidase 4.[2]

  1. ^ Beutner G, Sharma VK, Giovannucci DR, Yule DI, Sheu SS (June 2001). "Identification of a ryanodine receptor in rat heart mitochondria". The Journal of Biological Chemistry. 276 (24): 21482–8. doi:10.1074/jbc.M101486200. PMID 11297554.
  2. ^ Sun QA, Hess DT, Nogueira L, Yong S, Bowles DE, Eu J, Laurita KR, Meissner G, Stamler JS (September 2011). "Oxygen-coupled redox regulation of the skeletal muscle ryanodine receptor-Ca2+ release channel by NADPH oxidase 4". Proceedings of the National Academy of Sciences of the United States of America. 108 (38): 16098–103. Bibcode:2011PNAS..10816098S. doi:10.1073/pnas.1109546108. PMC 3179127. PMID 21896730.